Selection of papers on solid phase peptide synthesis published during 1996 to March 2001
- Balaspiri, L., & Langel, U. (2001) Synthesis of b-amyloid precursor peptide and presenilin segments. J. Peptide Sci., 7, 58-60. #16430
- Bullesbach, E.E., & Schwabe, C. (2001) Synthesis and conformational analysis of the insulin-like 4 gene product. J. Pept. Res., 57, 77-83. #16258
- Burgess, K., Han, I., Zhang, A., Zheng, W.H., Shanmugam, K., Featherstone, M.S., & Saragovi, H.U. (2001) DiSSiMiL: Diverse Small Size Mini-Libraries applied to simple and rapid epitope mapping of a monoclonal antibody. J. Pept. Res., 57, 68-76. #16259
- Dekker, N., Cox, R.C., Kramer, R.A., & Egmond, M.R. (2001) Substrate specificity of the integral membrane protease OmpT determined by spatially addressed peptide libraries. Biochemistry, 40, 1694-1701. #16271
- Demarcus, M., Ganadu, M.L., Mura, G.M., Porcheddu, A., Quaranta, L., Reginato, G., & Taddei, M. (2001) Small ring constrained peptidomimetics. Synthesis of epoxy peptidomimetics, inhibitors of cysteine proteases. J. Org. Chem., 66, 697-706. #16273
- Dolence, E.K., Dolence, J.M., & Poulter, C.D. (2001) Solid-phase synthesis of a radiolabeled, biotinylated, and farnesylated Ca(1)a(2)X peptide substrate for Ras- and a-mating factor converting enzyme. Bioconjug. Chem., 12, 35-43. #16275
- Futaki, S., Youjun, Z., & Sugiura, Y. (2001) Detecting a tag on a channel opening: Blockage of the biotinylated channels by strepravidin. Tetrahedron Lett., 42, 1563-1565. #16423
- Gatos, D., & Tzavara, C. (2001) Comparison of the solid-phase fragment condensation and phase-change approaches in the synthesis of salmon I calcitonin. J. Pept. Res., 57, 168-174. #16427
- Geginat, G., Schenk, S., Skoberne, M., Goebel, W., & Hof, H. (2001) A novel approach of direct ex vivo epitope mapping identifies dominant and subdominant CD4 and CD8 T cell epitopes from Listeria monocytogenes. Journal of Immunology, 166, 1877-1884. #16288
- Henlin, J.M., Boutin, J.A., Kucharczyk, N., Desmet-Beaufort, C., Loynel, A., Bertrand, M., Genton, A., Tucker, G.C., Atassi, G., & Fauchere, J.L. (2001) From peptide libraries to optimized nonpeptide ligands in the search for S-farnesyltransferase inhibitors. J. Pept. Res., 57, 85-96. #16425
- Kitagawa, K., Aida, C., Fujiwara, H., Yagami, T., Futaki, S., Kogire, M., Ida, J., & Inoue, K. (2001) Facile solid-phase synthesis of sulfated tyrosine-containing peptides: Total synthesis of human big gastrin-II and cholecystokinin (CCK)-39(1,2). J. Org. Chem., 66, 1-10. #16313
- Kumar, K.S., Roice, M., Sasikumar, P.G., Poduri, C.D., Sugunan, V.S., Pillai, V.N.R., & Das, M.R. (2001) Syntheses of immunodominant peptide regions of hepatitis C viral pathogens using PS-BDODMA resin: A single peptide derived from the conserved domain (E2/NS1) was highly effective in detecting anti-HCV antibodies. J. Pept. Res., 57, 140-150. #16426
- Lelievre, D., Bure, C., Laot, F., & Delmas, A. (2001) Synthesis of peptide di-aldehyde precursor for stepwise chemoselective ligations via oxime bonds. Tetrahedron Lett., 42, 235-238. #16326
- Licha, K., Hessenius, C., Becker, A., Henklein, P., Bauer, M., Wisniewski, S., Wiedenmann, B., & Semmler, W. (2001) Synthesis, characterization, and biological properties of cyanine-labeled somatostatin analogues as receptor-targeted fluorescent probes. Bioconjug. Chem., 12, 44-50. #16329
- Marchetto, R., Nicolas, E., Castillo, N., Bacardit, J., Navia, M., Vila, J., & Giralt, E. (2001) Two short peptides including segments of subunit A of Escherichia coli DNA gyrase as potential probes to evaluate the antibacterial activity of quinolones. J. Peptide Sci., 7, 27-40. #16441
- McNamara, L.M.A., Andrews, M.J.I., Mitzel, F., Siligardi, G., & Tabor, A.B. (2001) Unexpected conformational properties of a peptide constrained by an aliphatic link between the i and i+4 positions. Tetrahedron Lett., 42, 1591-1593. #16424
- Nilsson, M.R., Nguyen, L.L., & Raleigh, D.P. (2001) Synthesis and purification of amyloidogenic peptides. Anal. Biochem., 288, 76-82. #16355
- Qiu, W., Gu, X., Soloshonok, V.A., Carducci, M.D., & Hruby, V.J. (2001) Stereoselective synthesis of conformationally constrained reverse turn dipeptide mimetics. Tetrahedron Lett., 42, 145-148. #16181
- Royo, M., Jimenez, J.C., Lopez-Macia, A., Giralt, E., & Albericio, F. (2001) Solid-phase synthesis of peptides containing alpha,beta-didehydroamino acids. Eur. J. Org. Chem., 45-48. #16373
- Shuker, S.B., Esterbrook, J., & Gonzalez, J. (2001) Solid-phase synthesis of a novel peptide substituted calix[4]arene. Synlett, 210-213. #16382
- Aimoto, S., Hasegawa, K., Li, X. & Kawakami, T. (2000) Synthesis of phosphorylated CRE BP1(19-106) amide using a phosphopeptide thioester prepared directly by an Fmoc solid-phase method. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 82-83). Kluwer Academic Publisher, Dordrecht. #15701
- Ajikumar, P.K., & Devaky, K.S. (2000) EGDMA-cross-linked polystyrene resin: An efficient support for gel phase peptide synthesis. Proc. Indian Acad. Sci. -Chem. Sci., 112, 465-474. #15819
- Alam, M.R., Maeda, M., & Sasaki, S. (2000) DNA-binding peptides searched from the solid-phase combinatorial library with the use of the magnetic beads attaching the target duplex DNA. Bioorg. Med. Chem., 8, 465-473. #14913
- Albericio, F. (2000) Orthogonal protecting groups for Na-amino and C-terminal carboxyl functions in solid-phase peptide synthesis. Biopolymers (Pept. Sci. ), 55, 123-139. #16434
- Albericio, F. (2000) Orthogonal protecting groups for N alpha-amino and C-terminal carboxyl functions in solid-phase peptide synthesis. Biopolymers, 55, 123-139. #16237
- Alsina, J., Yokum, T.S., Albericio, F., & Barany, G. (2000) A modified Backbone Amide Linker (BAL) solid-phase peptide synthesis strategy accommodating prolyl, N-alkylamino acyl, or histidyl derivatives at the C-terminus. Tetrahedron Lett., 41, 7277-7280. #15629
- Alsina, J., Yokum, T.S., Albericio, F. & Barany, G. (2000) Backbone Amide Linker (BAL) methodology to accommodate C-terminal hindered, unreactive, and/or sensitive modification. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 102-103). Kluwer Academic Publisher, Dordrecht. #15707
- Andersson, L., Blomberg, L., Flegel, M., Lepsa, L., Nilsson, B., & Verlander, M. (2000) Large-scale synthesis of peptides. Biopolymers (Pept. Sci. ), 55, 227-250. #16440
- Andersson, L., Blomberg, L., Flegel, M., Lepsa, L., Nilsson, B., & Verlander, M. (2000) Large-scale synthesis of peptides. Biopolymers, 55, 227-250. #16238
- Ando, S., Nakahara, Y., Ito, Y., & Ogawa, T. (2000) Solid-phase synthesis of the glycopeptide of human glycophorin AM bearing the consecutive sialyl-T antigen. Carbohyd. Res., 329, 773-780. #16239
- Anichini, B., Ricci, R., Fabbri, G., Balacco, G., Mauro, S., Triolo, A., Altamura, M., Maggi, C.A., & Quartara, L. (2000) Solid-phase synthesis of MEN 11270, a new cyclic peptide kinin B2 receptor antagonist. J. Peptide Sci., 6, 612-620. #16152
- Annis, I. & Barany, G. (2000) Alternative solid-phase reagents for formation of intramolecular sulfur-sulfur bridges in peptides under mild conditions. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 96-97). Kluwer Academic Publisher, Dordrecht. #15704
- Antopolsky, M., & Azhayev, A. (2000) Stepwise solid-phase synthesis of peptide-oligonucleotide phosphorothioate conjugates employing Fmoc peptide chemistry. Tetrahedron Lett., 41, 9113-9117. #15823
- Arnon, R., Tarrab-Hazdai, R., & Steward, M. (2000) A mimotope peptide-based vaccine against Schistosoma mansoni: Synthesis and characterization. Immunology, 101, 555-562. #16245
- Arunan, C., & Pillai, V.N.R. (2000) Synthesis of acyl carrier protein fragment 65-74 on a flexible cross-linked polystyrene support: Comparison with Merrifield resin. Tetrahedron, 56, 3005-3011. #14623
- Arunan, C., Naaraj, R., & Pillai, V.N.R. (2000) Solid-phase synthesis of a modified 13-residue seminalplasmin fragment on 1,6-hexanediol diacrylate-crosslinked polystyrene support. Peptides, 21, 773-777. #15758
- Balaspiri, L., Tegyei, Z., Dux, M., Jancso, G., Jozsa, R., Csernus, V., & Mess, B. (2000) Synthesis of chicken galanin and its N- and C-terminal segments, and preparation of their antisera. Lett. Peptide Sci., 7, 23-26. #15431
- Balse, P., Han, G., Hruby, V.J. & Sun, L. (2000) Diisopropylethylamine salts for protected amino acids: Direct synthesis of peptides on solid-phase. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 80-81). Kluwer Academic Publisher, Dordrecht. #15700
- Balse, P.M., Kim, H.J., Han, G., & Hruby, V.J. (2000) Evaluation of new base-labile 2-(4-nitrophenylsulfonyl)ethoxycarbonyl (Nsc)-amino acids for solid-phase peptide synthesis. J. Pept. Res., 56, 70-79. #15444
- Baumann, M., Dietrich, U., Koenigs, C. & Griesinger, C. (2000) Combinatorial peptide synthesis, NMR-aided screening and testing of low molecular weight RNA-ligands. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 170-171). Kluwer Academic Publisher, Dordrecht. #15717
- Bechinger, B. (2000) Biophysical investigations of membrane perturbations by polypeptides using solid-state NMR spectroscopy. Molecular Membrane Biology, 17, 135-142. #15832
- Beebe, K.D., Wang, P., Arabaci, G., & Pei, D.H. (2000) Determination of the binding specificity of the SH2 domains of protein tyrosine phosphatase SHP-1 through the screening of a combinatorial phosphotyrosyl peptide library. Biochemistry, 39, 13251-13260. #15833
- Beligere, G.S., & Dawson, P.E. (2000) Design, synthesis, and characterization of 4-ester CI2, a model for backbone hydrogen bonding in protein alpha-helices. J. Amer. Chem. Soc., 122, 12079-12082. #16250
- Besser, D., Muller, B., Agricola, I., & Reissmann, S. (2000) Synthesis of differentially protected N-acylated reduced pseudodipeptides as building units for backbone cyclic peptides. J. Peptide Sci., 6, 130-138. #14943
- Besser, D., Muller, B., Kleinwachter, P., Greiner, G., Seyfarth, L., Steinmetzer, T., Arad, O., & Reissmann, S. (2000) Synthesis and characterization of octapeptide somatostatin analogues with backbone cyclization: Comparison of different strategies, biological activities and enzymatic stabilities. Journal fur Praktische Chemie-Practical Applications and Applied Chemistry, 342, 537-545. #15837
- Bibbs, L., Ambulos, N.P., Kates, S.A., Khatri, A., Medzihradszky, K.F., Osapay, G. & Weintraub, S.T. (2000) Strategies for the synthesis of labeled peptides. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 113-114). Kluwer Academic Publisher, Dordrecht. #15710
- Bishop, B.M., McCafferty, D.G., & Erickson, B.W. (2000) 4'-Aminomethyl-2,2'-bipyridyl-4-carboxylic acid (Abc) and related derivatives: Novel bipyridine amino acids for the solid-phase incorporation of a metal coordination site within a peptide backbone. Tetrahedron, 56, 4629-4638. #14946
- Blaskovich, M.A., Boatman, P.D., Cao, B., Eguchi, M., Kim, H.O., Lee, M., Little, T., Mathew, F., McCann, I., Mehlin, C., Nakanishi, H., Nelson, S., Nguyen, M., Ogbu, C., Qabar, M.N., Ruan, F., Shea, J.P., Stasiak, M., Urban, J. & Kahn, M. (2000) Highly efficient and versatile construction of secondary structure peptide mimetic libraries: Application to biology and drug development. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 191-193). Kluwer Academic Publisher, Dordrecht. #15726
- Blondelle, S.E., Crooks, E., Aligue, R., Agell, N., Bachs, O., Esteve, V., Tejero, R., Celda, B., Pastor, M.T., & Perez-Paya, E. (2000) Novel, potent calmodulin antagonists derived from an all-D hexapeptide combinatorial library that inhibit in vivo cell proliferation: Activity and structural characterization. J. Pept. Res., 55, 148-162. #14266
- Blondelle, S.E., Esteve, V., Celda, B., Pastor, M.T., & Perez-Paya, E. (2000) Influence of the hydrophylic face on the folding ability and stability of a-helix bundles: Relevance to the peptide catalytic activity. J. Pept. Res., 56, 121-131. #15789
- Bonner, G.G., Davis, P., Stropova, D., Edsall, S., Yamamura, H.I., Porreca, F., & Hruby, V.J. (2000) Opiate aromatic pharmacophore structure-activity relationships in CTAP analogues determined by topographical bias, two-dimensional NMR, and biological activity assays. J. Med. Chem., 43, 569-580. #14952
- Bordusa, F. (2000) Nonconventional amide bond formation catalysis: Programming enzyme specificity with substrate mimetics. Braz. J. Med. Biol. Res., 33, 469-485. #14953
- Borgia, J.A., Oegema, T.R.Jr. & Fields, G.B. (2000) Synthesis and application of a glycoprotein derived from the proteoglycan linkage structure. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 773-774). Kluwer Academic Publisher, Dordrecht. #15751
- Bourel, L., Carion, O., Gras-Masse, H., & Melnyk, O. (2000) The deprotection of Lys(Mtt) revisited. J. Peptide Sci., 6, 264-270. #14956
- Bourne, G.T., McGeary, R.P., Golding, S.W., Meutermans, W.D.F., Alewood, P.F. & Smythe, M.L. (2000) An evaluation of a novel safety catch linker for development of cyclic peptide libraries. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 98-99). Kluwer Academic Publisher, Dordrecht. #15705
- Boykins, R.A., Joshi, M., Syin, C., Dhawan, S., & Nakhasi, H. (2000) Synthesis and construction of a novel multiple peptide conjugate system: strategy for a subunit vaccine design. Peptides, 21, 9-17. #14958
- Boysen, R.I., & Hearn, M.T.W. (2000) Direct characterisation by electrospray ionisation mass spectroscopy of mercuro-polypeptide complexes after deprotection of acetamidomethyl groups from protected cysteine residues of synthetic polypeptides. J. Biochem. Biophys. Meth., 45, 157-168. #15846
- Bozo, B., Farkas, J., Toth, G., Wollemann, M., Szucs, M., & Benyhe, S. (2000) Receptor binding and G-protein activation by new Met(5)-enkephalin-Arg(6)-Phe(7) derived peptides. Life Sci., 66, 1241-1251. #14959
- Brask, J., & Jensen, K.J. (2000) Carbopeptides: Chemoselective ligation of peptide aldehydes to an aminooxy-functionalized D-galactose template. J. Peptide Sci., 6, 290-299. #15448
- Braslau, R., Axon, J.R., & Lee, B. (2000) Synthesis of N-hydroxy peptides: Chemical ligation of O-acyl hydroxamic acids. Organic Letters, 2, 1399-1401. #14964
- Buchardt, J., & Meldal, M. (2000) Novel methodology for the solid-phase synthesis of phosphinic peptides. Journal of the Chemical Society-Perkin Transaction 1, 3306-3310. #15852
- Bui, C.T., Ercole, F., Pham, Y., Campbell, R., Rasoul, F.A., Maeji, N.J., & Ede, N.J. (2000) Improving the performance of an acid-labile 4-hydroxymethyl phenoxyacetic acid (HMO) linker on resin and SynPhaseTM grafted solid-supports. J. Peptide Sci., 6, 534-538. #15756
- Bui, C.T., Bray, A.M., Nguyen, T., Ercole, F., Rasoul, F., Sampson, W., & Maeji, N.J. (2000) Acetophenone-based linker for solid-phase peptide synthesis. J. Peptide Sci., 6, 49-56. #14310
- Bui, C.T., Bray, A.M., Nguyen, T., Ercole, F., & Maeji, N.J. (2000) Solid phase synthesis of C-terminal peptide amides: Development of a new aminoethyl-polystyrene linker on the MultipinTM solid support. J. Peptide Sci., 6, 243-250. #14408
- Burgess, K. (2000) Solid-phase organic synthesis. John Wiley & Sons, New York. ISBN 0471318256 #14304
- Calcagni, A., Gavuzzo, E., Lucente, G., Mazza, F., Morera, E., Paradisi, M.P., & Rossi, D. (2000) Peptides containing the sulfonamide junction. 2. Structure and conformation of Z-Tau-Pro-D-Phe-NHiPr. Biopolymers, 54, 379-387. #15855
- Camarero, J.A., Adeva, A., & Muir, T.W. (2000) 3-Thiopropionic acid as a highly versatile multidetachable thioester resin linker. Lett. Peptide Sci., 7, 17-21. #15430
- Cammish, L.E., & Kates, S.A. (2000) Instrumentation for automated solid phase peptide synthesis. Fmoc Solid Phase Peptide Synthesis: A Practical Approaché, 222, 277-302. #15857
- Carlson, C.B., & Beal, P.A. (2000) Solid-phase synthesis of acridine-based threading intercalator peptides. Bioorg. Med. Chem. Lett., 10, 1979-1982. #15764
- Carreno, C., Mendez, M.E., Kim, Y.D., Kim, H.J., Kates, S.A., Andreu, D., & Albericio, F. (2000) Nsc and Fmoc Na-amino protection for solid-phase peptide synthesis: A parallel study. J. Pept. Res., 56, 63-69. #15443
- Cavero, M., Hobbs, A., Madge, D., Motherwell, W.B., Selwood, D., & Potier, P. (2000) Synthesis and biological evaluation of enantiopure thionitrites: The solid-phase synthesis and nitrosation of D-glutathione as a molecular probe. Bioorg. Med. Chem. Lett., 10, 641-644. #14632
- Cerovsky, V., & Bordusa, F. (2000) Protease-catalyzed fragment condensation via substrate mimetic strategy: A useful combination of solid-phase peptide synthesis with enzymatic methods. J. Pept. Res., 55, 325-329. #14363
- Chetyrkina, S., Estieu-Gionnet, K., Lain, G., Bayle, M., & Deleris, G. (2000) Synthesis of N-Fmoc-4-[(diethylphosphono)-2',2'-difluoro-1'-hydroxyethyl]phenylalanine, a novel phosphotyrosyl mimic for the preparation of signal transduction inhibitory peptides. Tetrahedron Lett., 41, 1923-1926. #14347
- Cho, J.K., Park, B.D., & Lee, Y.S. (2000) A novel core-shell type polymer support for solid-phase peptide synthesis. Tetrahedron Lett., 41, 7481-7485. #15861
- Cilli, E.M., Jubilut, G.N., Ribeiro, S.C.F., Oliveira, E., & Nakaie, C.R. (2000) Importance of the solvation degree of peptide-resin beads for amine groups determination by the picric acid method. J. Braz. Chem. Soc., 11, 474-478. #15862
- Clippingdale, A.B., Barrow, C.J., & Wade, J.D. (2000) Peptide thioester preparation by Fmoc solid phase peptide synthesis for use in native chemical ligation. J. Peptide Sci., 6, 225-234. #14405
- Conde-Frieboes, K., Andersen, S., & Breinholt, J. (2000) Synthesis of symmetrical dimeric N,N'-linked peptides on solid support by olefin metathesis. Tetrahedron Lett., 41, 9153-9156. #16159
- Cotton, G.J., & Muir, T.W. (2000) Generation of a dual-labeled fluorescence biosensor for Crk-II phosphorylation using solid-phase expressed protein ligation. Chem. Biol., 7, 253-261. #15864
- Cruz, L.J., Quintana, D., Iglesias, E., Garcia, Y., Huerta, V., Garay, H.E., Duarte, C., & Reyes, O. (2000) Immunogenicity comparison of a multi-antigenic peptide bearing V3 sequences of the human immunodeficiency virus type 1 with TAB9 protein in mice. J. Peptide Sci., 6, 217-224. #14402
- Cudic, M., Wade, J.D., & Otvos, L.Jr. (2000) Convenient synthesis of a head-to-tail cyclic peptide containing an expanded ring. Tetrahedron Lett., 41, 4527-4531. #14594
- Dai, X., Su, Z., & Liu, J.O. (2000) An improved synthesis of a selective aVb3-integrin antagonist cyclo(-RGDfK-). Tetrahedron Lett., 41, 6295-6298. #15531
- Dal, X.D., Su, Z., & Liu, J.O. (2000) An improved synthesis of a selective alpha(v)beta(3)-integrin antagonist cyclo(-RGDfK-). Tetrahedron Lett., 41, 6295-6298. #15868
- Dankwardt, S.M., Billedeau, R.J., Lawley, L.K., Abbot, S.C., Martin, R.L., Chan, C.S., Van Wart, H.E., & Walker, K.A.M. (2000) Solid-phase synthesis of di- and tripeptidic hydroxamic acids as inhibitors of procollagen C-proteinase. Bioorg. Med. Chem. Lett., 10, 2513-2516. #15870
- Denis, B., & Trifilieff, E. (2000) Synthesis of palmitoyl-thioester T-cell epitopes of myelin proteolipid protein (PLP). Comparison of two thiol protecting groups (StBu and Mmt) for on-resin-acylation. J. Peptide Sci., 6, 372-377. #15450
- Dionyssopoulou, H., Mouzaki, A., Slootstra, J., Puijk, W., Meloen, R., Cordopatis, P., & Sotiropoulou, G. (2000) Synthetic peptides as putative therapeutic agents in transplantation medicine: Application of PEPSCAN to the identification of functional sequences in the extracellular domain of the interleukin-2 receptor beta chain (IL-2R beta). J. Immunol. Method, 241, 83-95. #15882
- Dolence, E.K., Dolence, J.M., & Poulter, C.D. (2000) Solid-phase synthesis of a farnesylated CaaX peptide library: Inhibitors of the Ras CaaX endoprotease. Journal of Combinatorial Chemistry, 2, 522-536. #15605
- Drakopoulou, E., Uray, K., Mezo, G., Price, M.R., Vita, C., & Hudecz, F. (2000) Synthesis and antibody recognition of mucin 1 (MUC1)-a-conotoxin chimera. J. Peptide Sci., 6, 175-185. #14361
- Dufau, I., & Mazarguil, H. (2000) Design of a fluorescent amino acid derivative usable in peptide synthesis. Tetrahedron Lett., 41, 6063-6066. #15517
- Dutta, A.S., Gormley, J.J., Coath, M., Hassall, L., Hayward, C.F., Gellert, P.R., Kittlety, R.S., Alcock, P.J., Ferguson, R., Halterman, T., Jamieson, A., Moors, J.A., Moores, J.M., Rees, A., Wood, L.J., Reilly, C.F., & Haworth, D. (2000) Potent cyclic peptide inhibitors of VLA-4 (a4b1 integrin)-mediated cell adhesion. Discovery of compounds like cyclo(MePhe-Leu-Asp-Val-D-Arg-D-Arg) (ZD7349) compatible with depot formulation. J. Peptide Sci., 6, 398-412. #15453
- Dutta, A.S., Crowther, M., Gormley, J.J., Hassall, L., Hayward, C.F., Gellert, P.R., Kittlety, R.S., Alcock, P.J., Jamieson, A., Moores, J.M., Rees, A., Wood, L.J., Reilly, C.F., & Haworth, D. (2000) Potent cyclic monomeric and dimeric peptide inhibitors of VLA-4 (alpha(4)beta(1) integrin)-mediated cell adhesion based on the Ile-Leu-Asp-Val tetrapeptide. J. Peptide Sci., 6, 321-341. #15892
- Ede, N.J., Eagle, S.N., Wickham, G., Bray, A.M., Warne, B., Shoemaker, K., & Rosenberg, S. (2000) Solid phase synthesis of peptide aldehyde protease inhibitors. Probing the proteolytic sites of hepatitis C virus polyprotein. J. Peptide Sci., 6, 11-18. #13956
- Egleton, R.D., Mitchell, S.A., Huber, J.D., Janders, J., Stropova, D., Polt, R., Yamamura, H.I., Hruby, V.J., & Davis, T.P. (2000) Improved bioavailability to the brain of glycosylated Met-enkephalin analogs. Brain Res., 881, 37-46. #15894
- El-Agnaf, O.M.A., Mahil, D.S., Patel, B.P., & Austen, B.M. (2000) Oligomerization and toxicity of beta-amyloid-42 implicated in Alzheimer's disease. Biochem. Biophys. Res. Commun., 273, 1003-1007. #15895
- Falb, E., Yechezkel, T., Salitra, Y., Gellerman, G., Muller, D. & Gilon, C. (2000) In situ generation of Fmoc amino acid chlorides for extremely difficult couplings to sterically hindered secondary amines in solid-phase peptide synthesis. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 55-57). Kluwer Academic Publisher, Dordrecht. #15694
- Falchi, A., Giacomelli, G., Porcheddu, A., & Taddei, M. (2000) 4-(4,6-Dimethoxy[1,3,5]triazin-2-yl)-4-methyl-morpholinium chloride (DMTMM): A valuable alternative to PyBOP for solid phase peptide synthesis. Synlett, 275-277. #15026
- Fields, G.B., Tam, J.P., & Barany, G. (2000) Peptides for the New Millennium. Kluwer Academic Publisher, Dordrecht. ISBN 0792364457 #15688
- Fiertek, D., Gromowska, M., Andersen, A.R., Hansen, P.H., Majewski, T., & Izdebski, J. (2000) Primary structure of fox (Vulpes vulpes) proinsulin based on sequence studies of pancreatic peptides and cDNA. J. Peptide Sci., 6, 413-419. #15454
- Freund, E., Vitali, F., Linden, A., & Robinson, J.A. (2000) Solid-phase synthesis using (allyloxy)carbonyl(Alloc) chemistry of a putative heptapeptide intermediate in vancomycin biosynthesis containing m-chloro-3-hydroxytyrosine. Helv. Chim. Acta, 83, 2572-2579. #15902
- Fruchart, J.S., Grandjean, C., Bonnet, D., Rommens, C., Gras-Masse, H. & Melnyk, O. (2000) A new tartaric acid-based linker for the synthesis of C-terminal peptide a-oxo-aldehydes. In G.B. Fields, J.P. Tam & G. Barany (Eds.), Peptides for the New Millennium. (pp. 104-106). Kluwer Academic Publisher, Dordrecht. #15708
- Fruchart, J.S., Lippens, G., Warrass, R., Seetharaman, C., Dhalluin, C., & Boutillon, C. (2000) The Chemical Shift Index method applied to resin-bound peptides. J. Pept. Res., 56, 346-351. #16286
- Ghosh, A.K., & Fan, E. (2000) A novel method for sequence independent
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